What is Macimorelin?

The short answer

Macimorelin is a compound built to act like a peptide. In the US, you need a prescription to get Macimorelin.

Get updates on Macimorelin

What it is

Type
Ghrelin receptor agonist (oral peptidomimetic)
Also known as
macrilen
How it works
Stimulates GH release to test for GH deficiency.

Regulatory status

FDA-approved (Rx) How we label status

As of October 4, 2026, Macimorelin is an FDA-approved prescription drug for diagnosis of adult growth hormone deficiency.

See Macimorelin in the Index →

Federal (FDA)
Approved Rx (Macrilen NDA205598, 2017); Drugs@FDA lists Disc
503A compounding
Approved-drug component (not in any 503A category) (as of May 14, 2026)
WADA 2026
S2.2.4

References

Sources as of October 4, 2026

  1. DailyMed: dailymed.nlm.nih.gov/dailymed/drugInfo.cfm
  2. WADA: www.wada-ama.org/sites/default/files/2025-09/2026list_en_final_clean_september_2025.pdf